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Molecular association model of Peroxisome Proliferator-Activated Receptor α and its new specific and efficient ligand, K-877
- In: Poster Presentation
- At: Stockholm (Sweden) (2017)
- Type: Poster
- Poster code: P-A-075-Tuesday
- By: TOKIWA, Hiroaki (Rikkyo Universiry, Department of Chemistry, Tokyo, Japan)
- Co-author(s): Yurina Miyashita: Department of Chemistry, Rikkyo Universiry, Tokyo, Japan;AMED-CREST, JST, Tokyo, Japan
Kenta Takei: Department of Internal Medicine, University of Tsukuba, Tsukuba, Japan
Vladimir Sladek: Department of Chemistry, Rikkyo Universiry, Tokyo, Japan;AMED-CREST, JST, Tokyo, Japan
Shogo Nakano: Department of Food Sciences, University of Shizuoka, Shizuoka, Japan;AMED-CREST, JST, Tokyo, Japan
Shohei Ito: Department of Food Sciences, University of Shizuoka, Shizuoka, Japan;AMED-CREST, JST, Tokyo, Japan
Takeshi Matsuzaka: Department of Internal Medicine, University of Tsukuba, Tsukuba, Japan;AMED-CREST, JST, Tokyo, Japan
Motohiro Sekiya: Department of Internal Medicine, University of Tsukuba, Tsukuba, Japan;AMED-CREST, JST, Tokyo, Japan
Yoshimi Nakagawa: Department of Internal Medicine, University of Tsukuba, Tsukuba, Japan;AMED-CREST, JST, Tokyo, Japan
Hiroaki Tokiwa: Department of Chemistry, Rikkyo Universiry, Tokyo, Japan;AMED-CREST, JST, Tokyo, Japan
Hitoshi Shimano: Department of Internal Medicine, University of Tsukuba, Tsukuba, Japan;AMED-CREST, JST, Tokyo, Japan - Abstract:
Backgrounds
Peroxisome proliferator-activated receptors (PPARs) are ligand-activated transcription factors of nuclear receptor superfamily. PPARα is a regulator that activates fatty acid oxidation and improves hypertriglyceridemia. K-877 is a novel selective PPARα modulator (SPPARMα) to activate PPARα transcriptional activity.Aims
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Last update 28 September 2023