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Effects of CES1 genetic variants on its gene expression, and clopidogrel pharmacokinetics and pharmacodynamics
- In: Poster Presentation
- At: Stockholm (Sweden) (2017)
- Type: Poster
- Poster code: P-A-050-Tuesday
- By: NEUVONEN, Mikko (University of Helsinki, Clinical Pharmacology, Helsinki, Finland)
- Co-author(s): Mikko Neuvonen: Department of Clinical Pharmacology, University of Helsinki and Helsinki University Hospital, Helsinki, Finland
Katriina Tarkiainen: Department of Clinical Pharmacology, University of Helsinki and Helsinki University Hospital, Helsinki, Finland
Aleksi Tornio: Department of Clinical Pharmacology, University of Helsinki and Helsinki University Hospital, Helsinki, Finland
Päivi Hirvensalo: Department of Clinical Pharmacology, University of Helsinki and Helsinki University Hospital, Helsinki, Finland
Tuija Tapaninen: Department of Clinical Pharmacology, University of Helsinki and Helsinki University Hospital, Helsinki, Finland
Maria Paile-Hyvärinen: Department of Clinical Pharmacology, University of Helsinki and Helsinki University Hospital, Helsinki, Finland
Matti Itkonen: Department of Clinical Pharmacology, University of Helsinki and Helsinki University Hospital, Helsinki, Finland
Mikko Holmberg: Department of Clinical Pharmacology, University of Helsinki and Helsinki University Hospital, Helsinki, Finland
Vesa Kärjä: Department of Pathology, Kuopio University Hospital, Kuopio, Finland
Ville Männistö: Department of Medicine, University of Eastern Finland, Kuopio, Finland
Pertti Neuvonen: Department of Clinical Pharmacology, University of Helsinki and Helsinki University Hospital, Helsinki, Finland
Jussi Pihlajamäki: Department of Public Health and Clinical Nutrition, University of Eastern Finland, Kuopio, Finland;Clinical Nutrition and Obesity Center, Kuopio University Hospital, Kuopio, Finland
Janne Backman: Department of Clinical Pharmacology, University of Helsinki and Helsinki University Hospital, Helsinki, Finland
Mikko Niemi: Department of Clinical Pharmacology, University of Helsinki and Helsinki University Hospital, Helsinki, Finland - Abstract:
Backgrounds
Although carboxylesterase 1 (CES1) has a recognized role in drug metabolism and its activity shows marked interindividual variability, few studies have investigated the effects of genetic variants on CES1 expression in humans.
Aims
Our aim was to investigate effects of genetic variants on CES1 gene expression, and clopidogrel
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Last update 28 September 2023